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 2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole benzenesulfonate 2-(methylsulfonyl)-2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole Tert-butyl 6a-hydroxy-1,2,6,6a-tetrahydropyrrolo[3,4-c]pyrazole-5(4H)-carboxylate (Z)-tert-butyl 3-((dimethylamino)methylene)-4-oxopyrrolidine-1-carboxylate
 Tert-butyl 2-(methylsulfonyl)-4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole 4-methylbenzenesulfonate Tert-butyl 4,6-dihydropyrrolo[3,4-c]pyrazole-5(2H)-carboxylate (2S,3R,5S)-2-(2,5-difluorophenyl)-5-(2-(methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
 AZD8186 PRT-060318;PRT318 Omarigliptin;MK-3102 (R)-2-(2-methoxyphenyl)-2-((tetrahydro-2H-pyran-4-yl)oxy)ethanol
 BGB-324 BAR 502 (S)-2-amino-3-(4-fluoro-1H-indol-3-yl)propanoic acid CMS-024; YSL; alpha-BCP[7-9];Tyroserleutide
 H3B-6527 BAR 501 AP-26113 , Brigatinib CCT251545
 RTA-402; NSC-713200; TP-155C; Methyl-CDDO; MethylCDDO;Bardoxolone methyl OTS-964 CCT251921 BLU-9931
 (R)-methyl 5-(6-((4-methylpiperazin-1-yl)methyl)-1H-benzo[d]imidazol-1-yl)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate (R)-methyl 5-((5-((4-methylpiperazin-1-yl)methyl)-2-nitrophenyl)amino)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate (R)-methyl 5-amino-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate (R)-methyl 5-nitro-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxylate
 (S)-1-(2-(trifluoromethyl)phenyl)ethanol (S)-2-((1-(2-(trifluoromethyl)phenyl)ethoxy)carbonyl)benzoic acid (S)-1-phenylethanamine (S)-2-((1-(2-(trifluoromethyl)phenyl)ethoxy)carbonyl)benzoate 2-((1-(2-(trifluoromethyl)phenyl)ethoxy)carbonyl)benzoic acid
 1-(3-fluoro-4-nitrobenzyl)-4-methylpiperazine 3-fluoro-4-nitrobenzaldehyde 3-fluoro-N-methoxy-N-methyl-4-nitrobenzamide methyl 3-hydroxy-5-nitrothiophene-2-carboxylate
 methyl 3-hydroxythiophene-2-carboxylate GSK-461364A PZM-21 BLU-554
 Nazartinib; EGF816; NVS-816 (S)-2-((2-(1-isopropyl-1H-1,2,4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)oxy)propanamide TEW-7197; NOV-1301; EW-7197 3-(N-(4-methyl-2-nitro-5-(pyridin-3-yl)phenyl)sulfamoyl)benzoic acid
 (2-((5-chloro-2-((2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)amino)pyrimidin-4-yl)amino)phenyl)dimethylphosphine oxide 1-(4-fluoro-1H-indol-3-yl)-N-((R)-1-phenylethyl)propan-2-amine 1-(4-fluoro-1H-indol-3-yl)propan-2-one (E)-4-fluoro-3-(2-nitroprop-1-en-1-yl)-1H-indole
 4-fluoro-1H-indole-3-carbaldehyde (S)-1-(4-fluoro-1H-indol-3-yl)propan-2-amine (R)-1-(4-fluoro-1H-indol-3-yl)propan-2-amine tert-butyl ((3S,4S)-4-azidotetrahydro-2H-pyran-3-yl)carbamate
 (3R,4R)-3-((tert-butoxycarbonyl)amino)tetrahydro-2H-pyran-4-yl methanesulfonate tert-butyl ((3R,4R)-4-hydroxytetrahydro-2H-pyran-3-yl)carbamate (3R,4R)-3-(((R)-1-phenylethyl)amino)tetrahydro-2H-pyran-4-ol 3,7-dioxabicyclo[4.1.0]heptane
 3,6-dihydro-2H-pyran (3S,4S)-4-azidotetrahydro-2H-pyran-3-amine hydrochloride CB-5083 N-(5-((4-(1H-indol-3-yl)pyrimidin-2-yl)amino)-2-((2-(dimethylamino)ethyl)(methyl)amino)-4-methoxyphenyl)acrylamide
 (3aS,3bR,7aS,8aS)-2,2,5,5-tetramethyltetrahydro-3aH-[1,3]dioxolo[4’,5’:4,5]furo[3,2-d][1,3]dioxine 1H-inden-1-yl)-2-methylpropane-2-sulfinamide AMG-232 ACP-103; BVF-048;Nuplazid;Pimavanserin Tartrate
 GS-7340-03; TAF; Tenofovir Alafenamide Fumarate BEC HCl 4-(2-(4-((5,5-dimethyl-1,4,2-dioxathiolan-3-yl)methoxy)phenyl)propan-2-yl)phenol (1S,2R)-2-tert-Butoxycarbonylamino-cyclohexylamine
 (5-methylpyridin-2-yl)methyl acetate 3-[1-(4-bromobenzyl)-3-tert-butylsulfanyl-5-hydroxy-1H-indol-2-yl]-2,2-dimethylpropionic acid ethyl ester 5-[4-(bromomethyl)phenyl]-2-(ethyloxy)pyridine hydrobromide (R)-N-((R)-4-cyano-2,3-dihydro-1H-inden-1-yl)-2-methylpropane-2-sulfinamide
 (S)-tert-butyl (4-(5-(3-cyano-4-isopropoxyphenyl)-1,2,4-oxadiazol-3-yl)-2,3-dihydro-1H-inden-1-yl)carbamate S)-tert-butyl (2-((tert-butyldimethylsilyl)oxy)ethyl)(4-cyano-2,3-dihydro-1H-inden-1-yl)carbamate (S)-5-(3-(1-amino-2,3-dihydro-1H-inden-4-yl)-1,2,4-oxadiazol-5-yl)-2-isopropoxybenzonitrile 6-benzyloxy-8-((R)-2-chloro-1-hydroxy-ethyl)-4H-benzo[1,4]-oxazin-3-one
 2-(3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)azetidin-3-yl)acetonitrile tert-butyl 3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-(cyanomethyl)azetidine-1-carboxylate 4-((1,5-dimethyl-1H-pyrazol-3-yl)amino)-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxylic acid ethyl 4-amino-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxylate
 ethyl 1-ethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrrole-2-carboxylate 8-chloroisoquinolin-3-amine (R)-1-(dimethylamino)propan-2-ol 6-chloro-5-iodopyrazin-2-amine
 3,8-dichloroisoquinoline (R)-5-amino-3-((1-(dimethylamino)propan-2-yl)oxy)pyrazine-2-carbonitrile 5-amino-3-chloropyrazine-2-carbonitrile 6-chloropyrazin-2-amine
 SAR-020106 2-fluoro-2-methylpropan-1-ol (S)-tert-butyl (1-(1H-indol-3-yl)-3-iodopropan-2-yl)carbamate 2-fluoro-2-methylpropyl trifluoromethanesulfonate
 ethyl 2-fluoro-2-methylpropanoate (S)-tert-butyl (1-hydroxy-3-(1H-indol-3-yl)propan-2-yl)carbamate (E)-methyl 3-(3,5-difluoro-4-formylphenyl)acrylate 2-(4-bromo-2-chlorophenyl)acetic acid
 4-(ethylaMino)-2-(Methylthio)pyriMidine-5-carbaldehyde (R)-tert-butyl 3-(6-amino-8-oxo-7H-purin-9(8H)-yl)piperidine-1-carboxylate (R)-tert-butyl 3-(6-(dibenzylamino)-8-oxo-7H-purin-9(8H)-yl)piperidine-1-carboxylate (R)-tert-butyl 3-((5-amino-6-(dibenzylamino)pyrimidin-4-yl)amino)piperidine-1-carboxylate
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